API |
Product Name 產品名稱 |
CAS No. |
Structure 結構式 |
Patent 專利號 |
Rosuvastatin
瑞舒伐他汀鈣 |
Rosuvastatin methyl ester |
147118-40-9 |
 |
ZL200910053047.3
ZL201511022824.X
ZL201511022872.9
ZL201511023253.1
ZL201510940531.3 |
Rosuvastatin tert-butyl ester |
355806-00-7 |
 |
Tert-butyl 6-[(1E)-2-[4-(4-fluorophenyl)-6-(1-methylethyl)-2-[methyl(methylsulfonyl)amino]-5-pyrimidinyl]ethenyl]-2,2-dimethyl-1,3-dioxane-4-acetate |
289042-12-2 |
 |
Atorvastatin
阿托伐他汀鈣 |
4-Fluoro-α-(2-methyl-1-oxopropyl)-γ-oxo-N,β- diphenylbenzene butaneamide |
125971-96-2 |
 |
ZL200810202127.6 |
Diprotected Atorvastatin (L1) |
125971-95-1 |
 |
Perindopril
培哚普利 |
N-[(S)-1-Carbethoxybutyl]-(S)-alanine |
82834-12-6 |
 |
ZL201210555176.4
ZL200910266685.3 |
(S)-Indoline-2-carboxylic acid |
79815-20-6 |
 |
(2S,3aS,7aS)-Octahydro-1H-indole-2-carboxylic acid |
80875-98-5 |
 |
(2S,3aS,7aS)-Benzyl octahydro-1H-indole-2-carboxylate 4-methylbenzenesulfonate |
94062-52-9 |
 |
Ivabradine
伊伐布雷定 |
3-(3-Iodopropyl)-7,8-dimethoxy-1,3-dihydro-2H-3-benzapine-2-one |
148870-57-9 |
 |
ZL201010207206.3
ZL201510099954.7
ZL201511018565.3
|
[N-[[3,4-dimethoxybicyclo[4.2.0]octa-1,3,5-trien-7-yl] carbonyl]-N-methylamine] |
866783-13-3 |
 |
7,8-Dimethoxy-1,3-dihydro-2H-3-benzazepin-2-one |
73942-87-7 |
 |
Candesartan
坎地沙坦 |
Trityl candesartan |
139481-72-4 |
 |
ZL201010229921.7
ZL201510671739.X |
Ezetimibe
依替米貝 |
(4s)-3-[5-(4-Fluorophenyl)-1,5-dioxopenyl]-4-phenyl-2-oxazolidinone |
189028-93-1 |
 |
ZL201511030652.0 |
(S)-3-((S)-5-(4-Fluorophenyl)-5-hydroxypentanoyl)-4-phenyloxazolidin-2-one |
189028-95-3 |
 |
Methyl 3-[(2S,3R)-2-[4-(benzyloxy)phenyl]-1-(4-fluorophenyl)-4-oxoazetidin-3-yl]propanoate |
204589-80-0 |
 |
1-(4-Fluorophenyl)-3-[3-(4-fluorophenyl)-3-oxopropyl]-4-[4-(phenylmethoxy)phenyl]-(3R,4S)-2-azetidinone |
190595-65-4 |
 |
Galantamine
加蘭他敏 |
(+/-) Nawedine |
1668-86-6 |
 |
|
4a,5,9,10,11,12-Hexahydro-1-bromo-3-methoxy-11-formyl- 6H-Benzofuro[3a,3,2-ef][2] benzazepine-6-one |
122584-14-9 |
 |
Valsartan
纈沙坦 |
Methyl N-[(2’-Cyanobiphenyl-4-yl)methyl]-L-valinate hydrochloride |
482577-59-3 |
 |
ZL201010173862.6
ZL201510945518.7 |
Clopidogrel
氯吡格雷 |
(S)-Methyl (2-chlorophenyl)[(2-(2-thienyl)amino] acetate hydrochloride |
141109-19-5 |
 |
ZL201310462551.5 |
Pregabalin
普瑞巴林 |
(R)-(-)-3-(Carbamoylmethyl-5-methylmexanoic acid |
181289-33-8 |
 |
ZL201410137925.0
ZL201410675675.6 |
3-Carbamoymethyl-5-methylhexanoic acid |
181289-15-6 |
 |
Venlafaxine
文拉法辛 |
1-[2-Amino-1-(4-methoxyphenyl)-ethyl]-cyclohexanol |
130198-05-9 |
 |
ZL200910100326.0 |
Duloxetine
度洛西汀 |
(S)-3-(Methylamino)-1-(2-thienyl)-1-propanol |
116539-55-0 |
 |
ZL201410436429.5 |
S-(-)-N,N-Dimethyl-3-hydroxy-3-(2-thienyl)propanamine |
132335-44-5 |
 |
S-(+)-N,N-Dimethyl-3-(1-naphthoxy)-3-(2-thienyl)-1-propylamine oxalate |
132335-47-8 |
 |
Levocetirizine
左西替利嗪 |
(-)-1-[(4-Chlorophenyl) phenylmethyl]piperazine |
300543-56-0 |
 |
|
Donepezil
多奈哌齊 |
5,6-Dimethoxy-2-(4-piperidinylmet hyl)-1-indanone |
120014-30-4 |
 |
|
Dabigatran
達比加群 |
Ethyl 3-(4-(methylamino)-3-nitro-N-(pyridin-2-yl)benzamido)propanoate |
429659-01-8 |
 |
ZL201510411877.4
|
3-[(3-Amino-4-methylaminobenzoyl)pyridin-2-ylamino]propionic acid ethyl ester |
212322-56-0 |
 |
2-(4-Cyanophenylamino)acetic acid |
42288-26-6 |
 |
Ethyl 3-[[[2-[[(4-Cyanophenyl)amino]methyl]-1-methyl-1H-benzimidazol-5-yl]carbonyl]pyridin-2-ylamino] propionate |
211915-84-3 |
 |
N-[[2-[[[4-(Aminoiminomethyl)phenyl]amino]methyl]-1-methyl-1H-benzimidazol-5-yl]carbonyl]-N-2-pyridinyl-beta-alanine ethyl ester |
429658-95-7 |
 |
Ropinirole
羅匹尼羅 |
4-(2-Hydroxyethyl)-2H-indolin-2-one
|
139122-19-3
|
 |
|
Vildagliptin
維格列汀 |
(S)-1-(2-Chloroacetyl)pyrrolidine-2-carboxamide |
214398-99-9 |
 |
ZL201410112710.3 |
(2S)-1-(Chloroacetyl)-2-pyrrolidinecarbonitrile |
207557-35-5 |
 |
Dapagliflozin
達格列凈 |
5-Bromo-2-chloro-4’-ethoxydiphenylmethane |
461432-23-5 |
 |
ZL201510404207.X
|
Lesinurad
利拉利德 |
1-Cyclopropyl-4-isothiocyanatonaphthalene |
878671-95-5 |
 |
|
3H-1,2,4-Triazole-3-thione, 5-amino-4-(4-cyclopropyl-1-naphthalenyl)-2,4-dihydro |
878671-96-6 |
 |
Isopropyl 2-((5-bromo-4-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazol-3-yl)thio)acetate |
NA |
 |
Sitagliptin
西他列汀 |
5-[1-Hydroxy-2-(2,4,5-trifluorophenyl)ethylidene]-2,2-dimethyl-1,3-dioxane-4,6-dione |
767340-03-4 |
 |
|
(2Z)-4-Oxo-4-[3-(trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a]pyrazine-7(8H)-yl]-1-(2,4,5-trifluorophenyl)but-2-en-2-amine |
486460-32-6 |
 |
(3R)-3-Amino-1-[3-(trifluoromethyl)-5,6,7,8-tetrahydro-1,2,4-triazolo[4,3-a]pyrazin-7-yl]-4-(2,4,5-trifluorophenyl)butan-1-one |
486460-32-6 |
 |
Boc-(R)-3-Amino-4-(2,4,5-trifluorophenyl)butanoic acid |
486460-00-8 |
 |
Safinamide
沙芬酰胺 |
4-((3-Fluorobenzyl)oxy)benzaldehyde |
66742-57-2 |
 |
ZL201510952335.8 |
(S)-2((4-((3-Fluorobenzyl)oxy)benzyl)amino)propanamide |
133865-89-1 |
 |